An operationally simple procedure, involving conjugate addition of NaI to β-(2-aminophenyl)-α,β-ynones/cyclization/Pd-catalyzed reaction with 2-alkynyl-trifluoroacetanilides, afforded 4-(1H-indol-3-yl)quinolines. The whole process was carried out in the same flask, without any intermediate work-up and using ethanol as solvent.
A Concise One-Pot Approach to the Synthesis of 4-(1H-Indol-3-yl)quinolines
CHIARINI, MARCO;
2011-01-01
Abstract
An operationally simple procedure, involving conjugate addition of NaI to β-(2-aminophenyl)-α,β-ynones/cyclization/Pd-catalyzed reaction with 2-alkynyl-trifluoroacetanilides, afforded 4-(1H-indol-3-yl)quinolines. The whole process was carried out in the same flask, without any intermediate work-up and using ethanol as solvent.File in questo prodotto:
Non ci sono file associati a questo prodotto.
I documenti in IRIS sono protetti da copyright e tutti i diritti sono riservati, salvo diversa indicazione.
